Exemestane

Description

What is Aromasin (Exemestane)?

Exemestane is an orally active drug that is being used most often for treating breast cancer in women, but is also very famous for bodybuilding purposes for dealing with estrogenic related side effects. Exemestane is the active substance (chemical name) and is sold as the brand name Aromasin (brand for Exemestane) but is also found as many other trade names either.

Exemestane is an anti estrogen and more specifically is an aromatase inhibitor (AI). There are also SERMs in anti estrogens, but AIs and SERMs are highly different from each other, despite the fact that they are all working on inhibiting estrogen.

Aromatase Inhibitors (AIs) like Exemestane most commonly sold as Aromasin are blocking the synthesis of estrogen, as a result this is lowering the total estrogen levels in the body.

People who need to lower the estrogen levels (often due to hormonally breast cancer in medical settings or due to anabolic steroid use in bodybuilding communities) can use Exemestane with great success.

This drug has been approved by FDA back in 1999 and has become very popular all around the world for post menopausal women, but except for that – is very famous in bodybuilding as a way to prevent or treat estrogenic related side effects that may be induced from the use of steroids.

How Long Does Aromasin Stay in Your System? | Exemestane Half Life

Exemestane is staying in your system for twice as much as is the half life for this medication and taken in consideration that, according to scientists, it offers the half life of 25-27 hours, it stays in your system for at least 2 days and even a bit more.
You could use it once every other day or on a daily basis – no need for more frequent administration.

What is Aromasin (Exemestane) Used For in BodyBuilding?

In medical settings – Aromasin which is containing Exemestane as active substance is being used as an adjuvant treatment of post menopausal women that are having estrogen receptor positive early breast cancer. It is also given as treatment of advanced breast cancer and generally, the compound is used only for different needs when talking about hormonally positive breast cancer in women – cancers that require estrogen to grow.

In bodybuilding, Aromasin – Exemestane is used for blocking the synthesis of estrogen. This lowers the total amount of estrogen in the body and therefore allows the user to stay away from unwanted negative side effects related to too high levels of estrogen.

Too high estrogen levels can occur due to natural causes but it can artificially increase due to the use of anabolic steroids, those steroids that convert into estrogen known as aromatizable steroids also called “wet” steroids.

If a person uses such steroids, he might need Exemestane as a medicine to prevent or treat estrogen related side effects.

Exemestane is different from other AIs by not temporarily binding to the aromatase enzyme, but as soon as it binds – it stays there permanently. This means that Exemestane doesn’t have the risk of “estrogen rebound” as with other AIs that can occur after stopping their use.

Aromasin (Exemestane) Dosage in Bodybuilding

As it was already mentioned – Exemestane is an orally active drug which means that it should be taken orally by mouth. Due to its half life, Exemestane found in Aromasin or other trade names, is a medication that can be used once a day or once every other day.

If you’re getting prescribed Aromasin then use it exactly as your doctor told you to use it. By using it for bodybuilding purposes, then usually the dosage is dependent on the steroid type and dosage.

You do not need high dose of Exemestane when you use a low dosage of moderate aromatizable steroid. But you might need to increase the dosage of the AI if the dosage of a highly aromatizable steroid is increased.

Usually, a blood work determining the amount of estrogen in the body is best for determining the dosage of the drug. But most often, Exemestane is taken anywhere between 12.5 mg on and every other day basis up to about 25 mg on a daily basis (usually in the worst cases).

Do not use more than you need because this way you would inhibit too much estrogen and this comes with side effects.

Aromasin (Exemestane) Side Effects

Exemestane is a powerful aromatase inhibitor. This means that if you’re going to use too much Aromasin (or other trade names products containing Exemestane), then you would inhibit too much estrogen and this comes with negative side effects too. They can include:

• Loss of energy
• Loss of libido
• Loss of muscles
• Depression and various others

Side effects are mostly seen among female users and are rarely being reported among males. Nonetheless, sometimes they still report getting side effect of joint pain from dryness. Yet, this side effect and all other can be controlled and reduced by reducing the dosage.

Where to Buy Aromasin (Exemestane) for Men in Bodybuilding?

Exemestane can be purchased directly from this source and would offer a very high quality Exemestane 25 mg for bodybuilding purposes or for any other purposes when you need to lower down your estrogen levels.

Aromasin or other products containing high quality Exemestane would permanently bind to the aromatase enzyme and would lower the estrogen levels just enough for you to stay away from the negative side effects related to estrogen and avoid estrogen rebound.

https://medlineplus.gov/druginfo/meds/a607006.html
https://www.aromasin.com/
https://en.wikipedia.org/wiki/Exemestane
https://www.evolutionary.org/aromasin-exemestane